平安! 发表于 2011-11-9 19:57 + i; t/ @" M( q6 D- Q, V
Pazopanib (100 mg/kg/day free base equivalent) ' S9 N! h# O1 z, b& x N+ b
这是个已经在美国上市的老药了,能下载到正式药物使用说明书英文版。
/ J8 }& K3 H; N. J. Z搜索了一下,原料一大堆。
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对不起!100mg/kg是用于移植瘤的,我弄错了。2 l$ |; T' z3 ^1 N3 k
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以下是正版说明书的推荐用量。
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# v& n/ z9 q- H# I3 i--------------------- DOSAGE AND ADMINISTRATION ----------------* H- `! Z/ G% E; ~/ d7 d
* 800 mg orally once daily without food (at least 1 hour before or 2 hours after a meal). (2.1) . H& B$ @ S: X x; B
* Baseline moderate hepatic impairment – 200 mg orally once daily. Not recommended in patients with severe hepatic impairment. (2.2) 8 W* Z. l8 e" X
---------------------DOSAGE FORMS AND STRENGTHS --------------
) Q( ^' A9 t% W1 ?200 mg tablets. (3) : n8 D' O1 y- C/ v6 `9 M' Z
-------------------------------CONTRAINDICATIONS------------------------ |